✦ LIBER ✦

A New Synthesis of Sulfonamides by Aminolysis of p -Nitrophenylsulfonates Yielding Potent and Selective Adenosine A 2B Receptor Antagonists

✍ Scribed by Yan, Luo; Bertarelli, Daniela C. G.; Hayallah, Alaa M.; Meyer, Heiko; Klotz, Karl-Norbert; Müller, Christa E.

Book ID: 121371390
Publisher: American Chemical Society
Year: 2006
Tongue: English
Weight: 119 KB
Volume: 49
Category: Article
ISSN: 0022-2623
DOI: 10.1021/jm060277v

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

1,8-Disubstituted Xanthine Derivatives:

1,8-Disubstituted Xanthine Derivatives: Synthesis of Potent A 2B -Selective Adenosine Receptor Antagonists

✍ Hayallah, Alaa M.; Sandoval-Ramírez, Jesús; Reith, Ulrike; Schobert, Ulrike; Pre 📂 Article 📅 2002 🏛 American Chemical Society 🌐 English ⚖ 127 KB

Discovery of LAS101057: A Potent, Select

Discovery of LAS101057: A Potent, Selective, and Orally Efficacious A2B Adenosine Receptor Antagonist

✍ Eastwood, Paul; Esteve, Cristina; González, Jacob; Fonquerna, Silvia; Aiguadé, 📂 Article 📅 2010 🏛 American Chemical Society 🌐 English ⚖ 996 KB

Design, Synthesis, and Biological Evalua

Design, Synthesis, and Biological Evaluation of New 8-Heterocyclic Xanthine Derivatives as Highly Potent and Selective Human A 2B Adenosine Receptor Antagonists

✍ Baraldi, Pier Giovanni; Tabrizi, Mojgan Aghazadeh; Preti, Delia; Bovero, Andrea; 📂 Article 📅 2004 🏛 American Chemical Society 🌐 English ⚖ 278 KB

In vitro pharmacology of SCH 58261, a ne

In vitro pharmacology of SCH 58261, a new potent and selective A2a adenosine receptor antagonist

✍ C. Zocchi; E. Ongini; A. Conti; S. Ferrara; A. Negretti; S. Dionisotti 📂 Article 📅 1995 🏛 Elsevier Science 🌐 English ⚖ 159 KB

Rapid synthesis of [18F]SR46349B, a pote

Rapid synthesis of [18F]SR46349B, a potent and selective 5-HT2 receptor antagonist

✍ Pingzhong Tan; Joanna S. Fowler; Yu-Shin Ding; David J. Schlyer 📂 Article 📅 1995 🏛 John Wiley and Sons 🌐 French ⚖ 483 KB

## Abstract F‐18 labeled SR46349B, a highly potent and selective 5‐HT~2~ receptor antagonist, was synthesized as a potential radioligand for PET studies of brain 5‐HT~2~ receptors. Nucleophilic aromatic substitution of __trans__‐1‐(2‐nitrophenyl)‐3‐(4‐methoxymethoxyphenyl)‐2‐propenone (10) with NCA

Anilide Derivatives of an 8-Phenylxanthi

Anilide Derivatives of an 8-Phenylxanthine Carboxylic Congener Are Highly Potent and Selective Antagonists at Human A 2B Adenosine Receptors

✍ Kim, Yong-Chul; Ji, Xiao-duo; Melman, Neli; Linden, Joel; Jacobson, Kenneth A. 📂 Article 📅 2000 🏛 American Chemical Society 🌐 English ⚖ 130 KB