A new concise synthesis of nectrisine an
β
MichaΓ«l Bosco; Philippe Bisseret; Claire Bouix-Peter; Jacques Eustache
π
Article
π
2001
π
Elsevier Science
π
French
β 254 KB
The synthesis of new sugar-derived phosphonic acids from protected nectrisine is described. The key step is a highly stereoselective addition of a phosphonate anion to a sugar-derived dihydropyrrole to provide a versatile synthetic intermediate which can be functionalised in multiple ways.