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A new entry to [1,2,4]triazolo[1,5-a][1,4]benzodiazepin-6-onesvia intramolecular nitrilimine cycloaddition to the cyano group

✍ Scribed by Gianluigi Broggini; Luisa Garanti; Giorgio Molteni; Gaetano Zecchi

Publisher: Elsevier Science
Year: 1998
Tongue: French
Weight: 502 KB
Volume: 54
Category: Article
ISSN: 0040-4020
DOI: 10.1016/s0040-4020(98)00922-3

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✦ Synopsis

A series of [l,2.4]triazolo [l,5-al[l,4]benzodiazepin-6-ones of potential pharmacological interest have been synthesised by means of intramolecular nitrilimine cycloadditions to the cyano group.

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