𝔖 Bobbio Scriptorium
✦   LIBER   ✦

A general synthetic route towards bastadins. Part 1: Synthesis of the eastern part of bastadins 4–16

✍ Scribed by Elias A. Couladouros; Vassilios I. Moutsos

Publisher
Elsevier Science
Year
1999
Tongue
French
Weight
276 KB
Volume
40
Category
Article
ISSN
0040-4039

No coin nor oath required. For personal study only.

✦ Synopsis

A general synthetic route for the construction of the eastern part of the macrocyclic bastadins 4-16 is presented. The brominated biaryl ethers are synthesized using the iodonium salt method. The synthesis is accomplished within 18 steps in 15.5% overall yield.

📜 SIMILAR VOLUMES

A general synthetic route towards bastad
A general synthetic route towards bastadins. Part 2: Synthesis of the western part of bastadins 4–16, and fully functionalized macrocycle of bastadin 12
✍ Elias A. Couladouros; Vassilios I. Moutsos 📂 Article 📅 1999 🏛 Elsevier Science 🌐 French ⚖ 215 KB

A general synthetic route for the construction of the western part of the macrocyclic bastadins 4-16 is presented. The western and the eastern segments were coupled using the imidazolide of the corresponding acid. The bromine at position y2 may be added at this advanced step regiospecifically, stren

ChemInform Abstract: Towards a Versatile
ChemInform Abstract: Towards a Versatile Synthesis of Kainoids. Part 1. Introduction of the C-3 and C-4 Substituents.
✍ J. E. BALDWIN; S. J. BAMFORD; A. M. FRYER; M. P. W. RUDOLPH; M. E. WOOD 📂 Article 📅 2010 🏛 John Wiley and Sons ⚖ 32 KB 👁 2 views

Towards a Versatile Synthesis of Kainoids. Part 1. Introduction of the C-3 and C-4 Substituents. -Starting from trans-4-hydroxy-Lproline, an enamine alkylation is used for the stereospecific introduction of the C-3 substituent of acromelic acid analogues. For the introduction of C-4 aryl substituen

ChemInform Abstract: Progress Toward the
ChemInform Abstract: Progress Toward the Total Synthesis of Callipeltin A. Part 1. Asymmetric Synthesis of (3S,4R)-3,4-Dimethylglutamine.
✍ Bo Liang; Patrick J. Carroll; Madeleine M. Joullie 📂 Article 📅 2001 🏛 John Wiley and Sons ⚖ 30 KB 👁 2 views

## Abstract ChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 100 leading journals. To access a ChemInform Abstract of an article which was published elsewhere, please select a “Full Text” option. The original article is trackable v