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A facile synthesis of 3-substituted pipecolic acids, chimeric amino acids

✍ Scribed by Gergely M. Makara; Garland R. Marshall


Publisher
Elsevier Science
Year
1997
Tongue
French
Weight
247 KB
Volume
38
Category
Article
ISSN
0040-4039

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✦ Synopsis


Three protected 3-substituted pipecolic acid analogs were prepared as constrained chimeric amino acid building blocks. The concise synthetic route enables the synthesis of other derivatives with sidechaln functionality of amino acids as well.


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