𝔖 Bobbio Scriptorium
✦   LIBER   ✦

A convergent synthesis of 4-substituted 1,2,3,4-tetrahydroisoquinolin-1-ones

✍ Scribed by Nathalie Cholleton; Samir Z. Zard

Publisher
Elsevier Science
Year
1998
Tongue
French
Weight
223 KB
Volume
39
Category
Article
ISSN
0040-4039

No coin nor oath required. For personal study only.

πŸ“œ SIMILAR VOLUMES

Chemically-enabled synthesis of 1,2,3,4-
Chemically-enabled synthesis of 1,2,3,4-tetrahydroisoquinolin-1-ones
✍ Paul S. Humphries; Gayatri Balan; Bruce M. Bechle; Edward L. Conn; Kenneth J. Di πŸ“‚ Article πŸ“… 2009 πŸ› Elsevier Science 🌐 French βš– 412 KB

We have developed a number of efficient protocols for the facile synthesis of 1,2,3,4-tetrahydroisoquinolin-1-ones. This synthetic methodology allowed concise and efficient exploration of the SAR in all areas of the molecule. A number of these methods proved to be versatile, efficient and amenable t

Photochemical synthesis of 1,2,3,4-tetra
Photochemical synthesis of 1,2,3,4-tetrahydroisoquinolin-3-ones from N-chloroacetylbenzylamines
✍ Masaki Ikeda; Ken-ichi Hirao; Yohmei Okuno; Naganori Numao; Osamu Yonemitsu πŸ“‚ Article πŸ“… 1977 πŸ› Elsevier Science 🌐 French βš– 793 KB

When N-chloroacetyl-3-hydroxybenzylamine (37) in aqueous acetonitrile was irradiated, both ortho and para photocyclizations with reference to the OH group occurred to give 7-and 5 -hydroxy -3 -oxo -1,2,3,4tetrahydroisoquinolines ($2, 53). Similarly, 1 -methylisoquinoline derivatives (54, 55) were sy