✦ LIBER ✦

A convenient synthesis of 2-amino-2-oxazolines and their pharmacological evaluation at cloned human α adrenergic receptors

✍ Scribed by Wai C. Wong; Diana Wang; Carlos Forray; Pierre J.-J. Vaysse; Theresa A. Branchek; Charles Gluchowski

Publisher: Elsevier Science
Year: 1994
Tongue: English
Weight: 400 KB
Volume: 4
Category: Article
ISSN: 0960-894X
DOI: 10.1016/0960-894x(94)85032-1

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

Pharmacological evaluation of UK-14,304

Pharmacological evaluation of UK-14,304 analogs at cloned human α adrenergic receptors

✍ Yoon T. Jeon; Chi Luo; Carlos Forray; Pierre J.-J. Vaysse; Theresa A. Branchek; 📂 Article 📅 1995 🏛 Elsevier Science 🌐 English ⚖ 207 KB

Synthesis of 2-Amino-3-heteroaroylthioph

Synthesis of 2-Amino-3-heteroaroylthiophenes and Evaluation of Their Activity as Potential Allosteric Enhancers at the Human A1 Receptor.

✍ Pier Giovanni Baraldi; Maria Giovanna Pavani; John C. Shryock; Allan R. Moorman; 📂 Article 📅 2005 🏛 John Wiley and Sons ⚖ 16 KB 👁 2 views

## Thiophene derivatives R 0090 Synthesis of 2-Amino-3-heteroaroylthiophenes and Evaluation of Their Activity as Potential Allosteric Enhancers at the Human A1 Receptor. -The synthesis of a series of title compounds (III) by a known procedure is reported. The effect of substituents at positions 4

Synthesis and pharmacological evaluation

Synthesis and pharmacological evaluation of 5,6,7,8-tetrahydro-6-[propyl[2-(2-thienyl)ethyl]amino]-1,2-naphthalenediol: A novel non-selective dopamine-receptor agonist

✍ Swier Copinga; Durk Dijkstra; Jan B. de Vries; Cor J. Grol; Alan S. Horn 📂 Article 📅 2010 🏛 Elsevier Science 🌐 English ⚖ 788 KB

## Abstract Based on the hypothesis that simultaneous stimulation of dopamine D~1~ and ‐D~2~ receptors could be beneficial for the treatment of Parkinson's disease^7,13^, we prepared 5,6,7,8‐tetrahydro‐6‐[propyl[2‐(2‐thienyl)ethyl]amino]‐1,2‐naphthalenediol (PTAT. 4), the diol analogue of N‐0437 (3

A New Synthetic Approach of N-(4-Amino-2

A New Synthetic Approach of N-(4-Amino-2-methylquinolin-6-yl)-2-(4-ethylphenoxymethyl)benzamide (JTC-801) and Its Analogues and Their Pharmacological Evaluation as Nociceptin Receptor (NOP) Antagonists.

✍ Isabella Sestili; Anna Borioni; Carlo Mustazza; Andrea Rodomonte; Luciana Turche 📂 Article 📅 2005 🏛 John Wiley and Sons ⚖ 27 KB

## Abstract For Abstract see ChemInform Abstract in Full Text.

ChemInform Abstract: Medetomidine Analog

ChemInform Abstract: Medetomidine Analogues as α2-Adrenergic Ligands. Part 3. Synthesis and Biological Evaluation of a New Series of Medetomidine Analogues and Their Potential Binding Interactions with α2- Adrenoceptors Involving a “Methyl Pocket”.

✍ X. ZHANG; J. E. DE LOS ANGELES; M.-Y. HE; J. T. DALTON; G. SHAMS; L. LEI; P. N. 📂 Article 📅 2010 🏛 John Wiley and Sons ⚖ 32 KB 👁 1 views

Synthesis and Structure—Activity Relatio

Synthesis and Structure—Activity Relationships of Uracil Derived Human GnRH Receptor Antagonists: (R)-3-[2-(2-Amino)phenethyl]-1-(2,6-difluorobenzyl)-6-methyluracils Containing a Substituted Thiophene or Thiazole at C-5.

✍ Martin W. Rowbottom; et al. et al. 📂 Article 📅 2005 🏛 John Wiley and Sons ⚖ 198 KB 👁 2 views