9-Oxobenzomorphans. II. A versatile process for the synthesis of 9-oxo-6,7-benzomorphans
✍ Scribed by Kavadias, Gerry; Velkof, Stephan; Belleau, Bernard
- Book ID
- 121332021
- Publisher
- NRC Research Press
- Year
- 1979
- Tongue
- French
- Weight
- 325 KB
- Volume
- 57
- Category
- Article
- ISSN
- 0008-4042
- DOI
- 10.1139/v79-294
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📜 SIMILAR VOLUMES
The total synthesis of chiral ~~4,7-lactam1~ 4 has been accomplished starting from &acetoxyazetidinone. An independent route from methyl penicillanate has been used to test the efficiency of the foregoing synthesis. We recently reported (1) the skeletal conversion of penicillanic acid to (+)-2,2,5,
## Abstract (+)‐__N__‐[^11^C]‐Benzyl‐__N__‐normetazocine (1__S__,5__S__,9__S__‐(+)‐__cis__‐2‐[^11^C]‐benzyl‐2′‐hydroxy‐5,9‐dimethyl‐6,7‐benzomorphan), a potent and selective ligand for the σ receptor, was prepared by N‐benzylation of (+)‐__cis__‐__N__‐normetazocine with [α‐^11^C]‐benzyl iodide in e