✦ LIBER ✦

[3H]A-804598 ([3H]2-cyano-1-[(1S)-1-phenylethyl]-3-quinolin-5-ylguanidine) is a novel, potent, and selective antagonist radioligand for P2X7 receptors

✍ Scribed by Diana L. Donnelly-Roberts; Marian T. Namovic; Bruce Surber; Srirajan X. Vaidyanathan; Arturo Perez-Medrano; Ying Wang; William A. Carroll; Michael F. Jarvis

Book ID: 116785036
Publisher: Elsevier Science
Year: 2009
Tongue: English
Weight: 408 KB
Volume: 56
Category: Article
ISSN: 0028-3908
DOI: 10.1016/j.neuropharm.2008.06.012

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

2-[(3a R ,4 R ,5 S ,7a S )-5-{(1 S )-1-[

2-[(3a R ,4 R ,5 S ,7a S )-5-{(1 S )-1-[3,5-Bis(trifluoromethyl)phenyl]-2-hydroxyethoxy}-4-(2-methylphenyl)octahydro-2 H -isoindol-2-yl]-1,3-oxazol-4(5 H )-one: A Potent Human NK 1 Receptor Antagonist with Multiple Clearance Pathways

✍ Kassick, Andrew J.; Jiang, Jinlong; Bunda, Jaime; Wilson, David; Bao, Jianming; 📂 Article 📅 2013 🏛 American Chemical Society 🌐 English ⚖ 949 KB

Binding of [3H]MSX-2 (3-(3-hydroxypropyl

Binding of [3H]MSX-2 (3-(3-hydroxypropyl)-7-methyl-8-(m-methoxystyryl)-1-propargylxanthine) to rat striatal membranes — a new, selective antagonist radioligand for A2A adenosine receptors

✍ Christa E. Müller; Juris Maurinsh; Roland Sauer 📂 Article 📅 2000 🏛 Elsevier Science 🌐 English ⚖ 134 KB

Design and Synthesis of trans -3-(2-(4-(

Design and Synthesis of trans -3-(2-(4-((3-(3-(5-Methyl-1,2,4-oxadiazolyl))- phenyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyl-2,3,4,5-tetrahydro- 1 H -3-benzazepine (SB-414796): A Potent and Selective Dopamine D 3 Receptor Antagonist

✍ Macdonald, Gregor J.; Branch, Clive L.; Hadley, Michael S.; Johnson, Christopher 📂 Article 📅 2003 🏛 American Chemical Society 🌐 English ⚖ 211 KB

5-Amino-1-(2,6-dichloro-4-trifluoromethy

5-Amino-1-(2,6-dichloro-4-trifluoromethyl-phenyl)-3- [3H3]-methylsulfanyl-1H-pyrazole-4-carbonitrile (CTOM): Synthesis and Characterization of a Novel and Selective Insect GABA Receptor Radioligand.

✍ Sanath K. Meegalla; Dario Doller; Gary M. Silver; Nancy Wisnewski; Richard M. So 📂 Article 📅 2004 🏛 John Wiley and Sons ⚖ 109 KB

KF26777 (2-(4-bromophenyl)-7,8-dihydro-4

KF26777 (2-(4-bromophenyl)-7,8-dihydro-4-propyl-1H-imidazo[2,1-i]purin-5(4H)-one dihydrochloride), a new potent and selective adenosine A3 receptor antagonist

✍ Mayumi Saki; Hiroshi Tsumuki; Hiromi Nonaka; Junichi Shimada; Michio Ichimura 📂 Article 📅 2002 🏛 Elsevier Science 🌐 English ⚖ 210 KB

Physicochemical and biopharmaceutical ch

Physicochemical and biopharmaceutical characterization of endo-2-(8-methyl-8-azabicyclo[3.2.1]oct-3-yl)-2,3-dihydro-1H-benz[e]isoindol-1-one (CR3124) a novel potent 5-HT3 receptor antagonist

✍ Andrea Cappelli; Valter Travagli; Iacopo Zanardi; Maurizio Anzini; Gianluca Gior 📂 Article 📅 2006 🏛 John Wiley and Sons 🌐 English ⚖ 422 KB

The physicochemical and biopharmaceutical properties, such as pK a , crystal habit, water solubility, logD, molecular structure and dynamics, and membrane permeability of CR3124 (endo-2-(8-methyl-8-azabicyclo[3.2.1]oct-3-yl)-2,3-dihydro-1Hbenz[e]isoindol-1-one, a novel potent 5-HT 3 receptor antagon