(2S,3R)-1,2-epoxy-3-butanol. A useful synthon for the preparation of chiral 1,2-diols.
β Scribed by James D. White; Myung-chol Kang; Bernard G. Sheldon
- Publisher
- Elsevier Science
- Year
- 1983
- Tongue
- French
- Weight
- 185 KB
- Volume
- 24
- Category
- Article
- ISSN
- 0040-4039
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Some L-aspartylnorbornylamino alcohol derivatives were synthesized as potential peptide sweeteners. Of these compounds, 3-(~-aspartylamino)-l-(3-methyl-2-norbornyl)-2-butanol displays an excellent sweetness potency. By further synthesis of one diastereoisomer, (2R,3R)-3-(~-aspartylamino)-1-[(2S,3R)-