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[18F]-ET-1 a pet radioligand for the endothelin receptor system — radiochemistry, position of label and in vivo biodistribution

✍ Scribed by P. Johnström; N. G. Harris; T. D. Fryer; F. I. Aigbirhio; J. C. Clark; J. D. Pickard; A. P. Davenport

Book ID: 112132589
Publisher: John Wiley and Sons
Year: 2001
Tongue: French
Weight: 234 KB
Volume: 44
Category: Article
ISSN: 0022-2135
DOI: 10.1002/jlcr.25804401144

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## Abstract 4‐Fluoro‐__N__‐{2‐[4‐(6‐trifluoromethylpyridin‐2‐yl)piperazin‐1‐yl]ethyl}benzamide is a full 5‐HT~1A~ agonist with high affinity (__pK__~__i__~=9.3), selectivity and a __c__ log __P__ of 3.045. The corresponding PET radioligand 4‐[^18^F]fluoro‐__N__‐{2‐[4‐(6‐trifluoromethylpyridin‐2‐yl)