✦ LIBER ✦

1,4-Diacylpiperazine-2-(S)-[(N-aminoalkyl)carboxamides] as novel, potent substance P receptor antagonists.

✍ Scribed by Sander G. Mills; Mu Tsu Wu; Malcolm MacCoss; Richard J. Budhu; Conrad P. Dorn Jr.; Margaret A. Cascieri; Sharon Sadowski; Catherine D. Strader; William J. Greenlee

Book ID: 108476999
Publisher: Elsevier Science
Year: 1993
Tongue: English
Weight: 354 KB
Volume: 3
Category: Article
ISSN: 0960-894X
DOI: 10.1016/s0960-894x(01)80747-2

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

Synthesis of (1S,2R)-1-Phenyl-2- [(S)-1-

Synthesis of (1S,2R)-1-Phenyl-2- [(S)-1-aminoalkyl]-N,N-diethylcyclopropanecarboxamides as Novel NMDA Receptor Antagonists Having a Unique NMDA Receptor Subtype Selectivity.

✍ Satoshi Shuto; et al. et al. 📂 Article 📅 2010 🏛 John Wiley and Sons ⚖ 32 KB 👁 2 views

Benzodiazepine amidines: Novel, water-so

Benzodiazepine amidines: Novel, water-soluble 5-amino-1,4-benzodiazepin-2-one derivatives as potent CCKB receptor antagonists

✍ V.G. Matassa; G.A. Showell; S. Bourrain; J.G. Neduvelil; S.R. Fletcher; R. Baker 📂 Article 📅 1994 🏛 Elsevier Science 🌐 English ⚖ 238 KB

Asymmetric synthesis and biological eval

Asymmetric synthesis and biological evaluation of N-cyclohexyl-4-[1-(2,4-dichlorophenyl)-1-(p-tolyl)methyl]piperazine-1-carboxamide as hCB1 receptor antagonists

✍ Linghuan Gao; Min Li; Tao Meng; Hongli Peng; Xin Xie; Yongliang Zhang; Yu Jin; X 📂 Article 📅 2011 🏛 Elsevier Science 🌐 French ⚖ 493 KB

ChemInform Abstract: Asymmetric Synthesi

ChemInform Abstract: Asymmetric Synthesis and Biological Evaluation of N-Cyclohexyl-4- [1-(2,4-dichlorophenyl)-1-(p-tolyl)methyl]piperazine-1-carboxamide as hCB1 Receptor Antagonists.

✍ Linghuan Gao; Min Li; Tao Meng; Hongli Peng; Xin Xie; Yongliang Zhang; Yu Jin; X 📂 Article 📅 2012 🏛 John Wiley and Sons ⚖ 38 KB 👁 1 views

## Abstract Two enantiomers of the most potent racemic compounds in a series of recently discovered benzhydrylpiperazines are prepared using the Davis‐Ellmann‐type sulfonamide chemistry.

(+)-(2R,5S)-4-[4-Cyano-3-(trifluoromethy

(+)-(2R,5S)-4-[4-Cyano-3-(trifluoromethyl)phenyl]-2,5-dimethyl-N-[6-(trifluoromethyl)pyridin-3- yl]piperazine-1-carboxamide (YM580) as an Orally Potent and Peripherally Selective Nonsteroidal Androgen Receptor Antagonist1

✍ Kinoyama, Isao; Taniguchi, Nobuaki; Toyoshima, Akira; Nozawa, Eisuke; Kamikubo, 📂 Article 📅 2006 🏛 American Chemical Society 🌐 English ⚖ 300 KB

N,N-Dimethyl-[9-(arylsulfonyl)-2,3,4,9-t

N,N-Dimethyl-[9-(arylsulfonyl)-2,3,4,9-tetrahydro-1H-carbazol-3-yl]amines as novel, potent and selective 5-HT6 receptor antagonists

✍ Nirogi, Ramakrishna V.S.; Konda, Jagadishu Babu; Kambhampati, Ramasastry; Shinde 📂 Article 📅 2012 🏛 Elsevier Science 🌐 English ⚖ 579 KB