For a long time, C 2 -symmetric ligands were dominating in asymmetric catalysis. However, more recently it was found that in several metal-catalyzed processes non-symmetric mixed-donor bidentate P,N-ligands are superior to C 2 -symmetric P,P-or N,N-ligands. Especially phosphinooxazolines (PHOX ligan
12th Workshop of the Central European Division e.V. of the International Isotope Society
✍ Scribed by V. Snieckus; N. J. Geach; G. P. Randall; C. J. Winfield; A. Studer; A. C. Spivey; T. Jones; C. Noban; G. J. Ellames; A. Kohler; H. Wadsworth; J. Rieke-Zapp; S. Stone-Elander; J. Goehl; B. Perry; J. Windels; M. H. Marx; J. Krüger; B. Manmontri; G. Fels; F. Wüst; T. Kniess; R. Bergmann; P. Mäding; F. Füchtner; C. S. Hilger; M. Halks–Miller; R. Horuk; L. Matei; C. Postolache; V. Fugaru; E. Condac; A. Dinischiotu; M. Costache; L. Matei; C. Postolache; V. Fugaru; J. Atzrodt; V. Derdau
- Publisher
- John Wiley and Sons
- Year
- 2004
- Tongue
- French
- Weight
- 246 KB
- Volume
- 47
- Category
- Article
- ISSN
- 0022-2135
- DOI
- 10.1002/jlcr.896
No coin nor oath required. For personal study only.
✦ Synopsis
Abstract
V Snieckus [Queen's University, Canada]—The Directed Ortho Metalation—Cross Coupling Symbiosis in Aromatic Synthesis.
N Geach, GP Randall, CJ Winfield [Scynexis, UK]—Isotopically Labelled 4‐Formylimidazole.
A Studer [Marburg University, Germany]—New Concepts in Tin‐Free Radical Chemistry.
AC Spivey, C Noban [Imperial College London, UK]. T Jones [Sheffield University, UK], GJ Ellames, A Kohler [Sanofi‐Synthélabo, UK], H Wadsworth [Amersham Biosciences, UK]—Opportunities for Isotope Labelling via Solid Phase Synthesis with Organogermanium Linkers.
J Rieke‐Zapp [Aventis Pharma, Germany]—Optimization of Reaction Conditions on mg‐Scale by Use of Screening Devices.
S Stone‐Elander [Karolinska Institute, Sweden]—Rerouting Radiochemistry with Microwaves.
J Goehl, B Perry, D Leuck, J Windels, M Marx [EaglePicher Pharmaceutical, USA]—GMP and Radiolabelled Syntheses of Capsaicin.
J Krüger, B Manmontri, G Fels [Paderborn University, Germany]—H/D‐Exchange in Aromatic Systems Using Transition Metal Catalysis.
F Wüst, T Kniess, R Bergmann [Research Centre Rossendorf, Germany]—Synthesis of a ^11^C‐Labelled Nonsteroidal Glucocorticoid Receptor Ligand as Potential Radiotracer for Imaging Brain Glucocorticoid Receptors with Positron Emission Tomography (PET).
P Mäding, F Füchtner [Research Centre Rossendorf, Germany], CS Hilger [Schering AG, Germany]. M Halks‐Miller, R Horuk [Berlix Biosciences, USA]—^18^F‐Labelling of a Potent Nonpeptide CCR1 Antagonist for the Diagnosis of the Alzheimer's Disease.
L Matei, C Postolache, V Fugaru, E Condac, A Dinischiotu, M Costache [Bukarest University, Romania]—Use of [1,2‐^3^H] Testosterone in 5α‐ Reductase Enzymatic Activity Dosing in Dermal Fibroblast Cultures from Polycystic Ovarian Patients.
L Matei, C Postolache, V Fugaru [Bukarest University, Romania]—Synthesis and Stability Studies of Acyclovir Labelled with Tritium.
J Atzrodt, V Derdau [Aventis Pharma, Germany]—Studies on Directed Ortho‐Metalation (DoM) as Convenient Tool for the Synthesis of Labeled Compounds.
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