1,2-dihydro-3,1-benzoxazin-4-one and 4-H-1,2-dihydro-pyrido-[2,3-d]-[1,3]-oxazin-4-one derivatives as potential prodrugs: Part II: Hydrolysis

1,2-dihydro-3,1-benzoxazin-4-one and 4H-

1,2-dihydro-3,1-benzoxazin-4-one and 4H-1,2-dihydro-pyrido-[2,3-d]-[1,3]-oxazin-4-one derivatives as potential prodrugs: Part III: Permeability through excised human skin in vitro

✍ Gerhard Schwenker; Jianbing Chen 📂 Article 📅 1991 🏛 John Wiley and Sons 🌐 English ⚖ 283 KB

The percutaneous permeation characteristics of 6 potential prodrugs 2-7 in comparison with their parent drug mefenamic acid (1) in virro using excised human skin were studied. The results show that all potential prodrugs tested were at least 2.0 times as effective as mefenamic acid; compounds 2 and

ChemInform Abstract: The Preparation of

ChemInform Abstract: The Preparation of 2-Hydroxyethyl-2,3-dihydro-2H-1,4-benzoxazin-3(4H)-one Derivatives.

✍ R. F. FRECHETTE; M. J. BEACH 📂 Article 📅 2010 🏛 John Wiley and Sons ⚖ 29 KB

The Preparation of 2-Hydroxyethyl-2,3-dihydro-2H-1,4-benzoxazin-3(4H)-one Derivatives. -An effective strategy for the preparation of the title compounds (III), important intermediates in the synthesis of a series of novel antibacterial agents, is described. -(FRECHETTE, R. F.; BEACH,

ChemInform Abstract: Investigations of 4

ChemInform Abstract: Investigations of 4H-3,1-Benzoxazines. Part 13. Bromination of 1,2-Dihydro-4H-3,1-benzoxazines.

✍ E. V. GROMACHEVSKAYA; G. D. KRAPIVIN; V. E. ZAVODNIK; V. G. KUL'NEVICH 📂 Article 📅 2010 🏛 John Wiley and Sons ⚖ 30 KB

## Abstract ChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 100 leading journals. To access a ChemInform Abstract of an article which was published elsewhere, please select a “Full Text” option. The original article is trackable v

ChemInform Abstract: Reaction of 3-p-Tol

ChemInform Abstract: Reaction of 3-p-Toluoyl-1,2-dihydro-4H-pyrrolo(2,1-c)(1,4)benzoxazine- 1,2,4-trione with Benzylamine. Synthesis, Crystal and Molecular Structure of Z-3-(1-Benzyl-2-hydroxy-4,5-dioxo-2-p- tolyltetrahydropyrrol-3-idene)-3,4-dihydro-2H-1,4-benzoxazin-2-one.

✍ Z. G. ALIEV; A. N. MASLIVETS; I. V. MASHEVSKAYA; YU. S. ANDREICHIKOV; L. O. ATOV 📂 Article 📅 2010 🏛 John Wiley and Sons ⚖ 29 KB

## Abstract ChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 100 leading journals. To access a ChemInform Abstract of an article which was published elsewhere, please select a “Full Text” option. The original article is trackable v

ChemInform Abstract: Investigation in 4H

ChemInform Abstract: Investigation in 4H-3,1-Benzoxazine Series. Part 12. N-Substitution Reactions of 1,2-Dihydro-4H-3,1-benzoxazines.

✍ E. V. GROMACHEVSKAYA; T. P. KOSULINA; F. V. KVITKOVSKII; V. G. KUL'NEVICH 📂 Article 📅 2010 🏛 John Wiley and Sons ⚖ 32 KB 👁 1 views

On the Conformation of 1-Aryl-1,4-dihydr

On the Conformation of 1-Aryl-1,4-dihydro-3(2H)-isoquinolinones

✍ Jerzy L. Mokrosz; Marek T. Cegla; Edward Szneler 📂 Article 📅 1992 🏛 John Wiley and Sons 🌐 English ⚖ 365 KB