A series of 9-alkyl aromatic 8-carbolines was synthesized and evaluated as inhibitors of mitrochondrial monoamine oxidase. The possible existence of a hydrophobic or hydrophilic region on the enzyme was explored. Substitution of an electron-withdrawing group such as acetyl on N-9 position reduced t
✦ LIBER ✦
β-Carbolines as selective monoamine oxidase inhibitors:In vivoimplications
✍ Scribed by Vivette Glover; J. Liebowitz; Ines Armando; M. Sandler
- Publisher
- Springer
- Year
- 1982
- Tongue
- English
- Weight
- 575 KB
- Volume
- 54
- Category
- Article
- ISSN
- 1435-1463
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