The reactions of mono Boc-protected amino monocarboxylic acids with phosphoranylideneacetonitrile yield ylido nitriles which on ozonolysis at low temperature form labile a,b-diketo nitriles. These derivatives may be used in situ for reaction with diamines or related dinucleophiles to yield hetero de
α,β-Diketo Nitriles as Dielectrophiles. Formation of Heterocyclic Derivatives of Amino Acids.
✍ Scribed by Harry H. Wasserman; Yun Oliver Long; Jonathan Parr
- Publisher
- John Wiley and Sons
- Year
- 2003
- Weight
- 148 KB
- Volume
- 34
- Category
- Article
- ISSN
- 0931-7597
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✦ Synopsis
Abstract
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