Unexpected partial H1-receptor agonism of imidazole-type histamine H3-receptor antagonists lacking a basic side chain

Meta-Substituted Aryl(thio)ethers as Pot

Meta-Substituted Aryl(thio)ethers as Potent Partial Agonists (or Antagonists) for the Histamine H 3 Receptor Lacking a Nitrogen Atom in the Side Chain §

✍ Pelloux-Léon, Nadia; Fkyerat, Abdellatif; Piripitsi, Antonia; Tertiuk, Wasyl; Sc 📂 Article 📅 2004 🏛 American Chemical Society 🌐 English ⚖ 152 KB

ω-(Imidazol-4-yl)alkane-1-sulfonamides:

ω-(Imidazol-4-yl)alkane-1-sulfonamides: a new series of potent histamine H3 receptor antagonists

✍ Matthew J. Tozer; Ildiko M. Buck; Tracey Cooke; S.Barret Kalindjian; Michael J. 📂 Article 📅 2002 🏛 Elsevier Science 🌐 English ⚖ 168 KB

2-(4-Alkylpiperazin-1-yl)quinolines as a

2-(4-Alkylpiperazin-1-yl)quinolines as a New Class of Imidazole-Free Histamine H 3 Receptor Antagonists

✍ Zaragoza, Florencio; Stephensen, Henrik; Peschke, Bernd; Rimvall, Karin 📂 Article 📅 2005 🏛 American Chemical Society 🌐 English ⚖ 130 KB

ChemInform Abstract: ω-(Imidazol-4-yl)al

ChemInform Abstract: ω-(Imidazol-4-yl)alkane-1-sulfonamide: A New Series of Potent Histamine H3 Receptor Antagonists.

✍ Matthew J. Tozer; Ildiko M. Buck; Tracey Cooke; S. Barret Kalindjian; Michael J. 📂 Article 📅 2010 🏛 John Wiley and Sons ⚖ 38 KB 👁 1 views

## Abstract ChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 100 leading journals. To access a ChemInform Abstract of an article which was published elsewhere, please select a “Full Text” option. The original article is trackable v

ChemInform Abstract: Identification of a

ChemInform Abstract: Identification of a Novel, Orally Bioavailable Histamine H3 Receptor Antagonist (Ia) Based on the 4-Benzyl-(1H-imidazol-4-yl) Template.

✍ Robert Aslanian; et al. et al. 📂 Article 📅 2010 🏛 John Wiley and Sons ⚖ 29 KB 👁 2 views

## Abstract ChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 100 leading journals. To access a ChemInform Abstract of an article which was published elsewhere, please select a “Full Text” option. The original article is trackable v

Development of FUB 181, a Selective Hist

Development of FUB 181, a Selective Histamine H3-Receptor Antagonist of High Oral in Vivo Potency with 4-(?gv-(Arylalkyloxy)alkyl)-1H-imidazole Structure

✍ Holger Stark; Annette Hüls; Xavier Ligneau; Katja Purand; Heinz Pertz; Jean-Mich 📂 Article 📅 1998 🏛 John Wiley and Sons 🌐 English ⚖ 106 KB 👁 1 views