Tick Repellents II: N-substituted azacyclopentanones and azacyclopentenones

✍ Scribed by W. A. Skinner; U. Rosentreter; T. Elward

• Book ID: 102404473
• Publisher: John Wiley and Sons
• Year: 1983
• Tongue: English
• Weight: 325 KB
• Volume: 72
• Category: Article
• ISSN: 0022-3549
• DOI: 10.1002/jps.2600721131

✦ Synopsis

Several N-substituted azacyclopentanones and azacyclopentenones were synthesized and evaluated as repellents for the brown dog tick Rhipicephalus sanguineus. Several of these compounds were more effective in our test system than were the standard repellents, N,N-diethyl-m-toluamide and butopyranoxyl.

Keyphrases N-Substituted azacyclopentanones-synthesis, structure-activity relationships, evaluation as tick repellents N-Substituted azacyclopentenones-synthesis, structure-activity relationships, evaluation as tick repellents Tick repellents-potential, N-substituted azacyclopentanones and azacyclopentenones, synthesis 98c a 93% at 0.29 mg/cm2 and 63% at 0.19 mg/cm2. * 82% at 0.29 mg/cmZ and 47% at 0.19 mg/cm2. 77% at 0.29 rng/cm2 and 20% at 0.19 mg/cm2.