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Thermal cycloaddition reaction of xanthene-9-thione with allenes: An ESR study

✍ Scribed by J. Kamphuis; H. J. T. Bos; A. H. Huizer


Publisher
John Wiley and Sons
Year
1986
Tongue
English
Weight
820 KB
Volume
24
Category
Article
ISSN
0749-1581

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✦ Synopsis


During the parallel (2 + 2)-and (4 + 2)-cycloaddition reactions of aromatic thiones such as xanthene-9-thione with substituted allenes XCH=C==CH, (X = OR, SR, NMe,, Ph), a strong ESR signal is observed. This signal is associated with the (4 + 2)-cycloaddition reaction, affording thiopyran derivatives 3,1lb-dihydro-2-

Computer analyses of this signal made possible its identification as emanating from a 9-xanthenyl radical substituted at the 1-and 9-positions. The type of xanthenyl radical that is formed in the thermal reaction E rad or F rad depends on the nature of the substituent X at the allenic system H,C=C=CHX. This investigation shows that where X = Ph and M e 2 , xanthenyl radicals of structure E rud aEe produced, and where X = 0-t-Bu and S-t-Bu xanthenyl radicals of structure F rad are produced. It is striking that this production is so selective.

On irradiation (h > 254 nm), the production of xanthenyl radicals is enhanced. The conformation of xanthenyl radicals E rad and the role of E rad and F rad in the formation of addition products E and F are discussed.