✦ LIBER ✦

The serotonin 5-HT4 receptor: Part 3: Design and pharmacological evaluation of a new class of antagonists

✍ Scribed by K.-H. Buchheit; F. Klein; E. Klöppner; H.-J. Pfannkuche; H. Mattes

Publisher: Elsevier Science
Year: 1995
Tongue: English
Weight: 259 KB
Volume: 5
Category: Article
ISSN: 0960-894X
DOI: 10.1016/0960-894x(95)00434-u

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

Synthesis and Biological Evaluation of a

Synthesis and Biological Evaluation of a Novel Structural Type of Serotonin 5-HT3 Receptor Antagonists.

✍ Ramachandran Venkatesha Perumal; Radhakrishnan Mahesh 📂 Article 📅 2006 🏛 John Wiley and Sons ⚖ 13 KB

## Abstract ChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 200 leading journals. To access a ChemInform Abstract, please click on HTML or PDF.

Discovery of new anti-depressants from s

Discovery of new anti-depressants from structurally novel 5-HT3 receptor antagonists: Design, synthesis and pharmacological evaluation of 3-ethoxyquinoxalin-2-carboxamides

✍ Radhakrishnan Mahesh; Thangaraj Devadoss; Dilip Kumar Pandey; Shvetank Bhatt 📂 Article 📅 2011 🏛 Elsevier Science 🌐 English ⚖ 281 KB

A novel series of 3-ethoxyquinoxalin-2-carboxamides were designed as per the pharmacophoric requirements of 5-HT 3 receptor antagonist using ligand-based approach. The desired carboxamides were synthesized from the key intermediate, 3-ethoxyquinoxalin-2-carboxylic acid by coupling with appropriate a

Synthesis, conformational and pharmacolo

Synthesis, conformational and pharmacological study of new compounds as possible antagonists of the 5HT-3 receptor

✍ B. Whelan; I. Iriepa; E. Gálvez; A. Orjales; C. Berisa; A. Labeaga; A.G. García; 📂 Article 📅 1994 🏛 Elsevier Science 🌐 English ⚖ 253 KB

Pharmacological properties of dolasetron

Pharmacological properties of dolasetron, a potent and selective antagonist at 5-HT3 receptors

✍ Robert C. Miller; Martin Galvan; Maurice W. Gittos; Paul L. M. van Giersbergen; 📂 Article 📅 1993 🏛 John Wiley and Sons 🌐 English ⚖ 626 KB

Microwave Assisted Synthesis of 2-(4-Sub

Microwave Assisted Synthesis of 2-(4-Substituted piperazin-1-yl)-1,8-naphthyridine-3-carbonitrile as a New Class of Serotonin 5-HT3 Receptor Antagonists.

✍ Radhakrishnan Mahesh; Ramachandran Venkatesha Perumal; Pandi Vijaya Pandi 📂 Article 📅 2005 🏛 John Wiley and Sons ⚖ 18 KB 👁 1 views

Dopamine/Serotonin Receptor Ligands. Par

Dopamine/Serotonin Receptor Ligands. Part 4. Synthesis and Pharmacology of Novel 3-Benzazecines and 3-Benzazonines as Potential 5-HT2A and Dopamine Receptor Ligands.

✍ Hussein El-Subbagh; Thomas Wittig; Michael Decker; Sigurd Elz; Martin Nieger; Jo 📂 Article 📅 2003 🏛 John Wiley and Sons ⚖ 117 KB 👁 2 views