The novel N-substituted benztropine anal
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Ahmed A. Othman; Amy H. Newman; Natalie D. Eddington
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Article
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2008
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John Wiley and Sons
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English
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GA2-50 is a novel N-substituted benztropine analog with improved potency and selectivity for the dopamine transporter. The pharmacokinetic and pharmacodynamic properties of GA2-50 were characterized as a part of its preclinical evaluation as a substitute medication for cocaine abuse. In vitro transp