✦ LIBER ✦

The interaction of azelastine with human lung histamine H1, beta, and muscarinic receptor-binding sites

✍ Scribed by Casale, Thomas B.

Book ID: 119059467
Publisher: Elsevier Science
Year: 1989
Tongue: English
Weight: 774 KB
Volume: 83
Category: Article
ISSN: 1097-6825
DOI: 10.1016/0091-6749(89)90013-4

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

Interaction of histamine H2-receptor ant

Interaction of histamine H2-receptor antagonists with GABA and benzodiazepine binding sites in the CNS

✍ Joan M. Lakoski; George K. Aghajanian; Dorothy W. Gallager 📂 Article 📅 1983 🏛 Elsevier Science 🌐 English ⚖ 348 KB

Delineation of Receptor-Ligand Interacti

Delineation of Receptor-Ligand Interactions at the Human Histamine H1 Receptor by a Combined Approach of Site-Directed Mutagenesis and Computational Techniques – or – How to Bind the H1 Receptor

✍ Aldo Jongejan; Rob Leurs 📂 Article 📅 2005 🏛 John Wiley and Sons 🌐 English ⚖ 313 KB 👁 2 views

## Abstract Histamine H~1~ antagonists or “antihistamines” are one of the most prescribed drug families in Western countries. They exert their effect by binding to the histamine H~1~ receptor, a receptor belonging to the class of rhodopsin‐like G protein‐coupled receptors (GPCRs). In this review, t

Modelling of the binding site of the hum

Modelling of the binding site of the human m1 muscarinic receptor: Experimental validation and refinement

✍ Hélène Bourdon; Susanne Trumpp-Kallmeyer; Herman Schreuder; Jan Hoflack; Marcel 📂 Article 📅 1997 🏛 Springer Netherlands 🌐 English ⚖ 586 KB

Site-Directed Mutagenesis of the Histami

Site-Directed Mutagenesis of the Histamine H1-Receptor Reveals a Selective Interaction of Asparagine207 with Subclasses of H1-Receptor Agonists

✍ R. Leurs; M.J. Smit; C.P. Tensen; A.M. Terlaak; H. Timmerman 📂 Article 📅 1994 🏛 Elsevier Science 🌐 English ⚖ 426 KB

Histamine H1-Receptor Binding Sites in G

Histamine H1-Receptor Binding Sites in Guinea Pig Brain Membranes: Regulation of Agonist Interactions by Guanine Nucleotides and Cations

✍ Raymond S. L. Chang; Solomon H. Snyder 📂 Article 📅 1980 🏛 John Wiley and Sons 🌐 English ⚖ 630 KB

Characterization of the Histamine H 4 Re

Characterization of the Histamine H 4 Receptor Binding Site. Part 1. Synthesis and Pharmacological Evaluation of Dibenzodiazepine Derivatives

✍ Smits, Rogier A.; Lim, Herman D.; Stegink, Bart; Bakker, Remko A.; de Esch, Iwan 📂 Article 📅 2006 🏛 American Chemical Society 🌐 English ⚖ 183 KB