✦ LIBER ✦

The discovery of a potent orally efficacious indole androgen receptor antagonist through in vivo screening

✍ Scribed by James C. Lanter; James J. Fiordeliso; Weiqin Jiang; George F. Allan; Muh-Tsann Lai; Olivia Linton; Do Won Hahn; Scott G. Lundeen; Zhihua Sui

Book ID: 108074181
Publisher: Elsevier Science
Year: 2007
Tongue: English
Weight: 163 KB
Volume: 17
Category: Article
ISSN: 0960-894X
DOI: 10.1016/j.bmcl.2006.09.086

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

Discovery and Characterization of ML398,

Discovery and Characterization of ML398, a Potent and Selective Antagonist of the D 4 Receptor with in Vivo Activity

✍ Berry, Cynthia B.; Bubser, Michael; Jones, Carrie K.; Hayes, John P.; Wepy, Jame 📂 Article 📅 2014 🏛 American Chemical Society 🌐 English ⚖ 451 KB

SCH-C (SCH 351125), an orally bioavailab

SCH-C (SCH 351125), an orally bioavailable, small molecule antagonist of the chemokine receptor CCR5, is a potent inhibitor of HIV-1 infection in vitro and in vivo

✍ Strizki, J. M.; Xu, S.; Wagner, N. E.; Wojcik, L.; Liu, J.; Hou, Y.; Endres, M.; 📂 Article 📅 2001 🏛 National Academy of Sciences 🌐 English ⚖ 149 KB

3-[(2 R )-Amino-2-phenylethyl]-1-(2,6-di

3-[(2 R )-Amino-2-phenylethyl]-1-(2,6-difluorobenzyl)-5-(2-fluoro-3-methoxyphenyl)- 6-methylpyrimidin-2,4-dione (NBI 42902) as a Potent and Orally Active Antagonist of the Human Gonadotropin-Releasing Hormone Receptor. Design, Synthesis, and in Vitro and in Vivo Characterization

✍ Tucci, Fabio C.; Zhu, Yun-Fei; Struthers, R. Scott; Guo, Zhiqiang; Gross, Timoth 📂 Article 📅 2005 🏛 American Chemical Society 🌐 English ⚖ 170 KB