In vitro binding profile and radiosynthe
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Barbara Wenzel; Achim Hiller; Steffen Fischer; Dietlind Sorger; Winnie Deuther-C
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Article
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2011
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John Wiley and Sons
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French
⚖ 273 KB
## Abstract Radiolabeled vesamicol analogs are promising candidates as ligands for the vesicular acetylcholine transporter (VAChT) to enable __in vivo__ imaging of early cholinergic degenerations in brain. The 4‐fluorobenzoyl‐substituted azaspirovesamicol derivative FBASV is one out of six novel ve