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Synthetic Methods and Reactions. Part 106. Suppression of anchimerically assisted rearrangement products in the synthesis of α-fluorocarboxylic acids from α-amino acids with 48:52 (w/w) hydrogen fluoride/pyridine [1]

✍ Scribed by George A. Olah; G. K. Surya Prakash; Yah Li Chao


Publisher
John Wiley and Sons
Year
1981
Tongue
German
Weight
153 KB
Volume
64
Category
Article
ISSN
0018-019X

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✦ Synopsis


Abstract

Anchimerically assisted rearrangement, observed in the fluorination of some α‐amino acids with 70 : 30 (w/w) hydrogen fluoride/pyridine (by weight) in the presence of NaNO~2~, is substantially or fully suppressed by using the less acidic reagent 48 : 52 (w/w) hydrogen fluoride/pyridine.