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Synthesis of β-alanyl-arginyl-glycyl-phenylalanyl-phenyl-alanyl-typosine amide labelled with tritium or carbon-14

✍ Scribed by Nobuyoshi Hayashi; Takeo Kawakami; Kazuo Shinozaki; Mitsuhiro Wakimasu; Masahiko Fujino


Book ID
102370879
Publisher
John Wiley and Sons
Year
1978
Tongue
French
Weight
336 KB
Volume
14
Category
Article
ISSN
0022-2135

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✦ Synopsis


Abstract

The synthesis of β‐Ala‐Arg‐Gly‐Phe‐Phe‐Tyr‐NH~2~ labelled with tritium on the tyrosine residue or with carbon‐14 on the arginine residue is described. The tritium labelled compound VII was prepared in 49% radiochemical yield from L‐[3, 5‐^3^H] tyrosine and benzyloxycarbonyl‐β‐alanyl‐nitro‐arginyl‐glycyl‐phenylalanyl‐phenylalanine. The carbon‐14 labelled compound XVI was synthesized in 17% radiochemical yield from L‐[U‐^14^C]arginine and glycyl‐phenylalanyl‐phenylalanyl‐tyrosine amide.