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Synthesis of pyrimidines from 2-trichloromethyl-4-dimethylamino-1,3-diaza-1,3-butadienes and electron deficient acetylenes

✍ Scribed by Angel Guzmán; Moisés Romero; Francisco X. Talamás; Joseph M. Muchowski

Publisher
Elsevier Science
Year
1992
Tongue
French
Weight
204 KB
Volume
33
Category
Article
ISSN
0040-4039

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✦ Synopsis

2-Trichloromethyl-4-dimethylamino-1,3-diaza-l,3-butadienes(3),prepared from trichlomacetamidme(1) and amide acetals 2, readily react with electron d&ie.nt acetylenes 4 to give 2-trichloromethylpyrimidines 5.

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