Synthesis of pyrazolecarbonylaminopyridinecarboxamides as herbicides
β Scribed by John J. Parlow
- Book ID
- 102340354
- Publisher
- Journal of Heterocyclic Chemistry
- Year
- 1998
- Tongue
- English
- Weight
- 493 KB
- Volume
- 35
- Category
- Article
- ISSN
- 0022-152X
No coin nor oath required. For personal study only.
β¦ Synopsis
Abstract
Target compounds from a herbicide lead area, pyrazolecarboxamides, were selected and synthesized. These targets were chosen based on 1) βstructuralβ similarities of 2aβc with other known bleaching herbicides, and 2) the structure activity relationship previously established with analogs of the lead compound 2a. Syntheses of three target compounds were accomplished, two of which involved various transformations and regioselective additions with a pyridine nucleus to afford novel pyridine derivatives. These targets were tested in whole plant assays with the herbicidal data reported.
π SIMILAR VOLUMES
A number of 6-(4-phenoxyphenoxy)pyrimidines and triazines were synthesized and their herbicidal activity was measured. Compounds with the methoxy groups at the 2-and 4-positions on the pyrimidine and triazine rings exhibited high herbicidal activity. Introduction of a substituent into the 5position
A new series of the 0-pyrimidinylsalicylates was synthesized and their herbicidal activity was examined. Some of these compounds showed very strong herbicidal activity under pre-and post-emergent treatment conditions against various kinds of grass and broadleaf weeds. Among these compounds, 0-(4, 6d