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Synthesis of an Orthogonally-Protected Bifunctional Amino Acid for Conformationally Constrained Peptides

✍ Scribed by Martin J.I Andrews; Alethea B Tabor*

Publisher: Elsevier Science
Year: 1997
Tongue: French
Weight: 461 KB
Volume: 38
Category: Article
ISSN: 0040-4039
DOI: 10.1016/s0040-4039(97)00545-5

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✦ Synopsis

The asymmetricsynthesisof (2s, 9R)-2,9-diaminodecanedioic acid, rnthogomllyprotectedfor incorporationinto cyclicpeptidesby solid-phasesynthesis,is described.

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