Synthesis of a radiolabeled type A cholecystokinin receptor antagonist, (R)-N-pentyl-N-(4,5-di[3H]pentyl) Nα-(3-quinolinoyl)glutamic acid amide

Probes for narcotic receptor mediated ph

Probes for narcotic receptor mediated phenomena 22. (1) synthesis and characterization of optically pure [3H](+)-4-[(αR)-α-((2S, 5R)-4-propyl-2,5-dimethyl-1-piperazinyl)-3-methoxybenzyl]-N, N-diethylbenzamide, [3H]SNC 121, a novel high affinity and selective ligand for delta opioid receptors

✍ Silvia N. Calderon; Craig M. Bertha; J. Silvio Gutkind; Heng Xu; John S. Partill 📂 Article 📅 1996 🏛 John Wiley and Sons 🌐 French ⚖ 236 KB 👁 2 views

Probes for Narcotic Receptor Mediated Phenomena 22. (1) Synthesis and Characterization of Optically Pure [3 H I ( +)-4-1 ( a R)-a -( ( 2 s ,5 R ) -4 -P r o p y I -2 , 5 -d i m e t h y l -l -p i p e r e z i n y l ) -3 -m e t h o x y b e n z y l ] -~, ~-d i e t h y l b e n z a m i d e , [3H]SNC 121, a