## Abstract A straightforward synthesis of 2,6‐disubstituted piperidines bearing α‐amino acid side‐chains was developed. Synthesis was based on a Horner−Wadsworth−Emmons condensation of a β‐ketophosphonate derived from an α‐amino acid residue with a β‐homologated aldehyde of an __N__‐protected amin
Synthesis of 2,6-Disubstituted Piperidine-Bearing α-Amino Acid Side-Chains.
✍ Scribed by Damien Boeglin; Annie Heitz; Jean Martinez; Jean-Alain Fehrentz
- Publisher
- John Wiley and Sons
- Year
- 2003
- Weight
- 113 KB
- Volume
- 34
- Category
- Article
- ISSN
- 0931-7597
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Abstract
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