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Synthesis of 2-aminomethyl-4-phenyl-1-azabicyclo[2.2.1]heptanes via LiAlH4-induced reductive cyclization of 2-(4-chloro-2-cyano-2-phenylbutyl)aziridines and evaluation of their antimalarial activity

✍ Scribed by D’hooghe, Matthias; Vervisch, Karel; Törnroos, Karl W.; Verhaeghe, Tom; Desmet, Tom; Lategan, Carmen; Smith, Peter J.; Chibale, Kelly; De Kimpe, Norbert

Book ID: 120595823
Publisher: Elsevier Science
Year: 2013
Tongue: English
Weight: 441 KB
Volume: 23
Category: Article
ISSN: 0960-894X
DOI: 10.1016/j.bmcl.2012.12.029

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