✦ LIBER ✦

Synthesis and SAR studies of benzimidazole derivatives as melanin concentrating hormone receptor 1 (MCHR1) antagonists: Focus to detune hERG inhibition

✍ Scribed by Sasmal, Pradip K.; Sasmal, Sanjita; Abbineni, Chandrasekhar; Venkatesham, B.; Rao, P. Tirumala; Roshaiah, M.; Khanna, Ish; Sebastian, V. J.; Suresh, J.; Singh, Manvendra P.; Talwar, Rashmi; Shashikumar, Dhanya; Reddy, K. Harinder; Frimurer, Thomas M.; Rist, Øystein; Elster, Lisbeth; Högberg, Thomas

Book ID: 120388246
Publisher: The Royal Society of Chemistry
Year: 2011
Tongue: English
Weight: 239 KB
Volume: 2
Category: Article
ISSN: 2040-2503
DOI: 10.1039/c1md00015b

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

ChemInform Abstract: Design and Optimiza

ChemInform Abstract: Design and Optimization of Quinazoline Derivatives as Melanin Concentrating Hormone Receptor 1 (MCHR1) Antagonists. Part 2.

✍ Pradip K. Sasmal; et al. et al. 📂 Article 📅 2012 🏛 John Wiley and Sons ⚖ 22 KB

Design and Synthesis of Orally Efficacio

Design and Synthesis of Orally Efficacious Benzimidazoles as Melanin-Concentrating Hormone Receptor 1 Antagonists.

✍ Wen-Lian Wu; et al. et al. 📂 Article 📅 2006 🏛 John Wiley and Sons ⚖ 9 KB 👁 1 views

Design and synthesis of orally efficacio

Design and synthesis of orally efficacious benzimidazoles as melanin-concentrating hormone receptor 1 antagonists

✍ Wen-Lian Wu; Duane A. Burnett; Mary Ann Caplen; Martin S. Domalski; Chad Bennett 📂 Article 📅 2006 🏛 Elsevier Science 🌐 English ⚖ 131 KB

Synthesis and SAR study of pyrrolo[3,4-b

Synthesis and SAR study of pyrrolo[3,4-b]pyridin-7(6H)-one derivatives as melanin concentrating hormone receptor 1 (MCH-R1) antagonists

✍ Lim, Chae Jo; Kim, Ji Young; Lee, Byung Ho; Oh, Kwang-Seok; Yi, Kyu Yang 📂 Article 📅 2013 🏛 Elsevier Science 🌐 English ⚖ 466 KB

Discovery of Orally Efficacious Melanin-

Discovery of Orally Efficacious Melanin-Concentrating Hormone Receptor-1 Antagonists as Antiobesity Agents. Synthesis, SAR, and Biological Evaluation of Bicyclo[3.1.0]hexyl Ureas

✍ McBriar, Mark D.; Guzik, Henry; Shapiro, Sherry; Paruchova, Jaroslava; Xu, Ruo; 📂 Article 📅 2006 🏛 American Chemical Society 🌐 English ⚖ 245 KB

Synthesis, Structure–Activity Relationsh

Synthesis, Structure–Activity Relationship, and Pharmacological Studies of Novel Melanin-Concentrating Hormone Receptor 1 Antagonists 3-Aminomethylquinolines: Reducing Human Ether-a-go-go-Related Gene (hERG) Associated Liabilities

✍ Kasai, Shizuo; Kamata, Makoto; Masada, Shinichi; Kunitomo, Jun; Kamaura, Masahir 📂 Article 📅 2012 🏛 American Chemical Society 🌐 English ⚖ 567 KB