## Abstract 4‐[3‐[4‐(2‐Methoxyphenyl)piperazin‐1‐yl]propoxy]‐4‐aza‐tricyclo[5.2.1.02,6]dec‐8‐ene‐3,5‐dione (4), a potent and selective 5‐HT~1A~ agonist, was labeled by ^11^C‐methylation of the corresponding desmethyl analogue 3 with ^11^C‐methyl triflate. The precursor molecule 3 was synthesized fr
Synthesis and in vivo evaluation of a novel 5-HT1Areceptor agonist radioligand [O-methyl-11C]2-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-4-methyl-1,2,4-triazine-3,5(2H,4H)dione in nonhuman primates
✍ Scribed by J. S. Dileep Kumar; Jaya Prabhakaran; Vattoly J. Majo; Matthew S. Milak; Shu-Chi Hsiung; Hadassah Tamir; Norman R. Simpson; Ronald L. Van Heertum; J. John Mann; Ramin V. Parsey
- Publisher
- Springer
- Year
- 2007
- Tongue
- English
- Weight
- 363 KB
- Volume
- 34
- Category
- Article
- ISSN
- 0340-6997
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