✦ LIBER ✦

Synthesis and in Vitro Evaluation of N-Substituted Maleimide Derivatives as Selective Monoglyceride Lipase Inhibitors

✍ Scribed by Matuszak, Nicolas; Muccioli, Giulio G.; Labar, Geoffray; Lambert, Didier M.

Book ID: 115450569
Publisher: American Chemical Society
Year: 2009
Tongue: English
Weight: 996 KB
Volume: 52
Category: Article
ISSN: 0022-2623
DOI: 10.1021/jm900461w

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

Design, Synthesis, and Biochemical Evalu

Design, Synthesis, and Biochemical Evaluation of N -Substituted Maleimides as Inhibitors of Prostaglandin Endoperoxide Synthases †

✍ Kalgutkar, Amit S.; Crews, Brenda C.; Marnett, Lawrence J. 📂 Article 📅 1996 🏛 American Chemical Society 🌐 English ⚖ 613 KB

Synthesis of Bicyclic N-Arylmethyl-Subst

Synthesis of Bicyclic N-Arylmethyl-Substituted Iminoribitol Derivatives as Selective Nucleoside Hydrolase Inhibitors

✍ Maya Berg; Gunther Bal; Annelies Goeminne; Pieter Van der Veken; Wim Versées; Ja 📂 Article 📅 2009 🏛 John Wiley and Sons 🌐 English ⚖ 510 KB

## Abstract **A series of bicyclic** **__N__****‐arylmethyl‐substituted iminoribitols** were synthesised and evaluated in vitro against __T. vivax__ nucleoside hydrolase. The importance of the N–Asp40 interaction was confirmed and depends on an optimal p__K__~a~ value, which can be influenced by su

Design, synthesis, and evaluation of (E)

Design, synthesis, and evaluation of (E)-N-substituted benzylidene–aniline derivatives as tyrosinase inhibitors

✍ Bae, Sung Jin; Ha, Young Mi; Park, Yun Jung; Park, Ji Young; Song, Yu Min; Ha, T 📂 Article 📅 2012 🏛 Elsevier Science 🌐 French ⚖ 542 KB

Synthesis and Evaluation of Substituted

Synthesis and Evaluation of Substituted Chroman-4-one and Chromone Derivatives as Sirtuin 2-Selective Inhibitors

✍ Fridén-Saxin, Maria; Seifert, Tina; Landergren, Marie Rydén; Suuronen, Tiina; La 📂 Article 📅 2012 🏛 American Chemical Society 🌐 English ⚖ 436 KB

ChemInform Abstract: Design, Synthesis,

ChemInform Abstract: Design, Synthesis, and Biochemical Evaluation of N-Substituted Maleimides as Inhibitors of Prostaglandin Endoperoxide Synthases (PGHS) .

✍ A. S. KALGUTKAR; B. C. CREWS; L. J. MARNETT 📂 Article 📅 2010 🏛 John Wiley and Sons ⚖ 31 KB

Synthesis and Pharmacological Evaluation

Synthesis and Pharmacological Evaluation of 2,4-Dinitroaryldithiocarbamate Derivatives as Novel Monoacylglycerol Lipase Inhibitors

✍ Kapanda, Coco N.; Masquelier, Julien; Labar, Geoffray; Muccioli, Giulio G.; Poup 📂 Article 📅 2012 🏛 American Chemical Society 🌐 English ⚖ 858 KB