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Synthesis, and conformational and biological study of 2-D-Ala,5-des-Met-enkephalin hydrazide modified at the carboxylic end by poly-N-vinylimidazole

✍ Scribed by G. Vlasov; E. Krasnikova; N. Kozhevnikova; N. Illarionova; I. Denisov


Publisher
Wiley (John Wiley & Sons)
Year
1987
Tongue
English
Weight
535 KB
Volume
26
Category
Article
ISSN
0006-3525

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✦ Synopsis


Synopsis

N, N-bis-2-~-Ala,5-des-Met-enkephalin hydrazide of azo-isobutyric acid was synthesized. This was used to obtain polyvinylimidazole derivatives of an enkephalin analog, modified at the carboxylic end by poly-N-vinylimidazole. The effect of modification of tetrapeptide hydrazide on its conformational properties and biological activity in viw and in vitro was studied.

*This paper is dedicated to the 70th anniversary of Professor G. Maneke.