## Abstract Iodocaramiphen (2) is a selective muscarinic antagonist which binds __in vitro__ with high affinity and selectivity to the M~1~ subtype of the muscarinic receptor. We report the synthesis of iodine‐125 labeled iodocaramiphen ([^125^I]‐2) via a tributylstannyl intermediate (3) in 50% rad
Synthesis and biological evaluation of125I-nebivolol as a potential cardioselective agent for imaging β1-adrenoceptors
✍ Scribed by M. A. Motaleb; M. E. Moustapha; I. T. Ibrahim
- Book ID
- 106442040
- Publisher
- Springer
- Year
- 2011
- Tongue
- English
- Weight
- 453 KB
- Volume
- 289
- Category
- Article
- ISSN
- 1588-2780
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