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Synthesis and biological evaluation of conformationally restricted derivatives of tryptophan as NK1/NK2 ligands

✍ Scribed by Régis Millet; Jean-François Goossens; Karine Bertrand-Caumont; Philippe Chavatte; Raymond Houssin; Jean-Pierre Hénichart

Book ID
110268674
Publisher
Springer Netherlands
Year
1999
Tongue
English
Weight
197 KB
Volume
6
Category
Article
ISSN
1573-3149

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Synthesis of New 4-Heteroaryl-2-Phenylqu
Synthesis of New 4-Heteroaryl-2-Phenylquinolines and Their Pharmacological Activity as NK-2/NK-3 Receptor Ligands
✍ Anna Borioni; Carlo Mustazza; Isabella Sestili; Maria Sbraccia; Luciana Turchett 📂 Article 📅 2007 🏛 John Wiley and Sons 🌐 English ⚖ 923 KB

## Abstract Substituted 4‐heteroaryl‐2‐phenylquinolines were synthesized and tested on NK‐2 and NK‐3 receptors in order to get a better insight in the structure‐activity relationship. On the whole, these molecules, which can be regarded as bioisosters of the NK‐3 antagonist SB 218795, displayed a l