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Synthesis and Biological Evaluation of 3-Heterocyclyl-7,8,9,10-tetrahydro-(7,10-ethano)-1,2,4-triazolo[3,4- a ]phthalazines and Analogues as Subtype-Selective Inverse Agonists for the GABA A α5 Benzodiazepine Binding Site

✍ Scribed by Street, Leslie J.; Sternfeld, Francine; Jelley, Richard A.; Reeve, Austin J.; Carling, Robert W.; Moore, Kevin W.; McKernan, Ruth M.; Sohal, Bindi; Cook, Susan; Pike, Andrew; Dawson, Gerard R.; Bromidge, Frances A.; Wafford, Keith A.; Seabrook, Guy R.; Thompson, Sally A.; Marshall, George; Pillai, Goplan V.; Castro, José L.; Atack, John R.; MacLeod, Angus M.

Book ID: 121858244
Publisher: American Chemical Society
Year: 2004
Tongue: English
Weight: 273 KB
Volume: 47
Category: Article
ISSN: 0022-2623
DOI: 10.1021/jm0407613

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