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Synthesis and Biological Characterization of Amidopropenyl Hydroxamates as HDAC Inhibitors

✍ Scribed by Florian Thaler; Mario Varasi; Andrea Colombo; Roberto Boggio; Davide Munari; Nickolas Regalia; Marco G. Rozio; Veronica Reali; Anna E. Resconi; Antonello Mai; Stefania Gagliardi; Giulio Dondio; Saverio Minucci; Ciro Mercurio

Book ID: 102105342
Publisher: John Wiley and Sons
Year: 2010
Tongue: English
Weight: 351 KB
Volume: 5
Category: Article
ISSN: 1860-7179
DOI: 10.1002/cmdc.201000166

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## Abstract The histone deacetylases (HDACs) are able to regulate gene expression, and inhibitors of the HDACs (HDACIs) hold promise in the treatment of cancer as well as a variety of neurodegenerative diseases. To investigate the potential for isoform selectivity in the inhibition of HDACs, we pre