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Synthesis and binding affinity of cis-(−)- and cis-(+)-N-ethyleneamino-N-nordeoxymetazocine and cis-(−)-N-normetazocine analogues at σ1, σ2 and κ opioid receptors

✍ Scribed by Giuseppe Ronsisvalle; Orazio Prezzavento; Agostino Marrazzo; Franco Vittorio; Ennio Bousquet; Rosanna Di Toro; Santi Spampinato

Book ID: 114301792
Publisher: Elsevier Science
Year: 2001
Tongue: English
Weight: 146 KB
Volume: 12
Category: Article
ISSN: 0928-0987
DOI: 10.1016/s0928-0987(00)00157-3

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## Abstract (+)‐__N__‐[^11^C]‐Benzyl‐__N__‐normetazocine (1__S__,5__S__,9__S__‐(+)‐__cis__‐2‐[^11^C]‐benzyl‐2′‐hydroxy‐5,9‐dimethyl‐6,7‐benzomorphan), a potent and selective ligand for the σ receptor, was prepared by N‐benzylation of (+)‐__cis__‐__N__‐normetazocine with [α‐^11^C]‐benzyl iodide in e