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Syntheses of 2-spiroindoles and pyrrolof[1,2-a]indoles

✍ Scribed by B. Malapel-Andrieu; J.-Y. Mérour

Publisher
Journal of Heterocyclic Chemistry
Year
1998
Tongue
English
Weight
543 KB
Volume
35
Category
Article
ISSN
0022-152X

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✦ Synopsis

Abstract

C‐alkylated products obtained from methyl 3‐hydroxyindole‐2‐carboxylate afford either spiro compounds, such as an indolic analogue of nitramine, or tricyclic products with a pyrrolo[1,2‐a]indole framework. Di‐C‐alkylated derivatives give access to tetracyclic compounds.

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