✦ LIBER ✦

Substitution of arginine for cysteine 643 of the glucocorticoid receptor reduces its steroid-binding affinity and transcriptional activity

✍ Scribed by Michiyo Nagano; Takahiro Nakamura; Shingo Niimi; Tomofumi Fujino; Tetsuji Nishimura; Norie Murayama; Seiichi Ishida; Shogo Ozawa; Yoshiro Saito; Jun-ichi Sawada

Book ID: 117467309
Publisher: Elsevier Science
Year: 2002
Tongue: English
Weight: 95 KB
Volume: 181
Category: Article
ISSN: 0304-3835
DOI: 10.1016/s0304-3835(02)00042-3

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

Steroid derivatives for electrophilic af

Steroid derivatives for electrophilic affinity labelling of glucocorticoid binding sites: Interaction with the glucocorticoid receptor and biological activity

✍ Alessandro Weisz; Robert L. Buzard; Diane Horn; Ming P. Li; Lois V. Dunkerton; F 📂 Article 📅 1983 🏛 Elsevier Science 🌐 English ⚖ 887 KB

Affinity of corticosteroids for mineralo

Affinity of corticosteroids for mineralocorticoid and glucocorticoid receptors of the rabbit kidney: Effect of steroid substitution

✍ M.E. Rafestin-Oblin; M. Lombes; P. Lustenberger; P. Blanchardie; A. Michaud; G. 📂 Article 📅 1986 🏛 Elsevier Science 🌐 English ⚖ 849 KB

Binding affinities of mometasone furoate

Binding affinities of mometasone furoate and related compounds including its metabolites for the glucocorticoid receptor of rat skin tissue

✍ Isogai, Mitsutaka; Shimizu, Hitoshi; Esumi, Yoshio; Terasawa, Tadao; Okada, Tosh 📂 Article 📅 1993 🏛 Elsevier Science 🌐 English ⚖ 325 KB

2-Substituted 5-methoxy-N-acyltryptamine

2-Substituted 5-methoxy-N-acyltryptamines: synthesis, binding affinity for the melatonin receptor, and evaluation of the biological activity

✍ Spadoni, Gilberto; Stankov, Bojidar; Duranti, Andrea; Biella, Gabriele; Lucini, 📂 Article 📅 1993 🏛 American Chemical Society 🌐 English ⚖ 719 KB

Peroxisome proliferator-activated recept

Peroxisome proliferator-activated receptor α and its response element are required but not sufficient for transcriptional activation of the mouse heart-type fatty acid binding protein gene

✍ Kowhei Kawabe; Hirokazu Saegusa; Kohichi Seto; Hiroaki Urabe; Kiyoto Motojima 📂 Article 📅 2005 🏛 Elsevier Science 🌐 English ⚖ 206 KB

Polymorphisms in the GATA-Binding Sites

Polymorphisms in the GATA-Binding Sites of the Vitamin D Receptor Gene Affect Its Transcription in the Esophagus, and Are Associated With a Reduced Risk for Esophageal Disease

✍ van de Winkel, Anouk ;Uitterlinden, André ;Rygiel, Agnieszka M. ;Moons, Leon M. 📂 Article 📅 2011 🏛 Elsevier Science 🌐 English ⚖ 64 KB