## Abstract This article describes in detail the first total synthesis of grandisine alkaloids, grandisines B, D, and F, which show affinity for the human δ‐opioid receptor. The key steps in this synthesis are construction of the isoquinuclidinone moiety of **2** by intramolecular imine formation a
✦ LIBER ✦
Studies Toward the Total Synthesis of Grandisine A: Synthesis of 9-epi-Grandisine A.
✍ Scribed by David J. Maloney; Samuel J. Danishefsky
- Publisher
- John Wiley and Sons
- Year
- 2007
- Weight
- 20 KB
- Volume
- 38
- Category
- Article
- ISSN
- 0931-7597
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