✦ LIBER ✦

Structure–activity relationship of a series of non peptidic RGD integrin antagonists targeting α5β1: Part 2

✍ Scribed by Bénédicte Delouvrié; Katherine Al-Kadhimi; Jean-Claude Arnould; Simon T. Barry; Darren A.E. Cross; Myriam Didelot; Paul R. Gavine; Hervé Germain; Craig S. Harris; Adina M. Hughes; David A. Jude; Jane Kendrew; Christine Lambert-van der Brempt; Jean-Jacques Lohmann; Morgan Ménard; Andrew A. Mortlock; Martin Pass; Claire Rooney; Michel Vautier; Jennifer L. Vincent; Nicolas Warin

Book ID: 113496883
Publisher: Elsevier Science
Year: 2012
Tongue: English
Weight: 830 KB
Volume: 22
Category: Article
ISSN: 0960-894X
DOI: 10.1016/j.bmcl.2012.04.061

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

Non-Peptide αvβ3 Antagonists. Part 5. Id

Non-Peptide αvβ3 Antagonists. Part 5. Identification of Potent RGD Mimetics Incorporating 2-Aryl β-Amino Acids as Aspartic Acid Replacements.

✍ Karen M. Brashear; et al. et al. 📂 Article 📅 2003 🏛 John Wiley and Sons ⚖ 88 KB

New non-peptide angiotensin II receptor

New non-peptide angiotensin II receptor antagonists. 2: structure - activity relationship of a series of annelated 2(1H)-pyridinones

✍ John R. Bantick; Haydn G. Beaton; Sally L. Cooper; Stephen Hill; Simon C. Hirst; 📂 Article 📅 1994 🏛 Elsevier Science 🌐 English ⚖ 396 KB

Synthesis and structure-activity relatio

Synthesis and structure-activity relationships of a novel series of non-peptide AT2-selective angiotensin II receptor antagonists

✍ M.T. Wu; T.J. Ikeler; W.T. Ashton; R.S.L. Chang; V.J. Lotti; W.J. Greenlee 📂 Article 📅 1993 🏛 Elsevier Science 🌐 English ⚖ 443 KB

Structure–activity relationship studies

Structure–activity relationship studies of a series of peptidomimetic ligands for α4 β1 integrin on Jurkat T-leukemia cells

✍ Ruiwu Liu; Li Peng; Huijun Han; Kit S. Lam 📂 Article 📅 2006 🏛 Wiley (John Wiley & Sons) 🌐 English ⚖ 357 KB

## Abstract α~4~β~1~ integrin is a therapeutic target for inflammation, autoimmune diseases, and lymphoid cancers. A series of peptidomimetic ligands based on the Nle‐D‐I motif have been synthesized and their binding affinities (IC~50~) to activated α~4~β~1~ integrin on Jurkat T‐leukemia cells have

Structure−Activity Relationship Studies

Structure−Activity Relationship Studies on a Series of Novel, Substituted 1-Benzyl-5-phenyltetrazole P2X 7 Antagonists

✍ Nelson, Derek W.; Gregg, Robert J.; Kort, Michael E.; Perez-Medrano, Arturo; Voi 📂 Article 📅 2006 🏛 American Chemical Society 🌐 English ⚖ 134 KB

Structure−Activity Relationships of a Se

Structure−Activity Relationships of a Series of Substituted Benzamides: Potent D 2 /5-HT 2 Antagonists and 5-HT 1a Agonists as Neuroleptic Agents

✍ Norman, Mark H.; Rigdon, Greg C.; Hall, William R.; Navas, Frank 📂 Article 📅 1996 🏛 American Chemical Society 🌐 English ⚖ 368 KB