✦ LIBER ✦

Structure-Affinity Relationships of Adenosine A2B Receptor Ligands

✍ Scribed by Margot W. Beukers; Illiana Meurs; Adriaan P. IJzerman

Publisher: John Wiley and Sons
Year: 2006
Weight: 8 KB
Volume: 37
Category: Article
ISSN: 0931-7597
DOI: 10.1002/chin.200647254

No coin nor oath required. For personal study only.

✦ Synopsis

Abstract

ChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 200 leading journals. To access a ChemInform Abstract, please click on HTML or PDF.

📜 SIMILAR VOLUMES

8-Substituted-9-deazaxanthines as Adenos

8-Substituted-9-deazaxanthines as Adenosine Receptor Ligands: Design, Synthesis and Structure-Affinity Relationships at A2B.

✍ Angelo Carotti; Angela Stefanachi; Enrique Ravina; Eddy Sotelo; Maria Isabel Loz 📂 Article 📅 2005 🏛 John Wiley and Sons ⚖ 13 KB

Structure-Affinity Relationships of the

Structure-Affinity Relationships of the Affinity of 2-Pyrazolyl Adenosine Analogues for the Adenosine A2A Receptor.

✍ Venkata P. Palle; Elfatih O. Elzein; Scott A. Gothe; Zhihe Li; Zhenhai Gao; Step 📂 Article 📅 2003 🏛 John Wiley and Sons ⚖ 72 KB 👁 1 views

Potent antagonists for the human adenosi

Potent antagonists for the human adenosine A2B receptor. Derivatives of the triazolotriazine adenosine receptor antagonist ZM241385 with high affinity

✍ Maarten de Zwart; Roel C. Vollinga; Margot W. Beukers; Danielle F. Sleegers; Jac 📂 Article 📅 1999 🏛 John Wiley and Sons 🌐 English ⚖ 147 KB 👁 2 views

A series of novel and known 5-substituted 7-amino-2-(2-furyl) [1,2,4]triazolo [1,5a][1,3,5]triazine derivatives were synthesized and tested for adenosine receptor antagonism in radioligand binding assays at all four adenosine receptor subtypes and for inhibition of the agonist-induced cyclic AMP res

ChemInform Abstract: Synthesis and Bindi

ChemInform Abstract: Synthesis and Binding Affinity of Homologated Adenosine Analogues as A3 Adenosine Receptor Ligands.

✍ Hyuk Woo Lee; Won Jun Choi; Kenneth A. Jacobson; Lak Shin Jeong 📂 Article 📅 2011 🏛 John Wiley and Sons ⚖ 29 KB 👁 1 views

The Discovery of a Selective, High Affin

The Discovery of a Selective, High Affinity A2B Adenosine Receptor Antagonist for the Potential Treatment of Asthma.

✍ Jeff Zablocki; et al. et al. 📂 Article 📅 2005 🏛 John Wiley and Sons ⚖ 27 KB 👁 2 views

Structural Predictions of Adenosine 2B A

Structural Predictions of Adenosine 2B Antagonist Affinity Using Molecular Field Analysis

✍ Song, Yuqing ;Coupar, Ian M. ;Iskander, Magdy N. 📂 Article 📅 2001 🏛 John Wiley and Sons 🌐 English ⚖ 515 KB