𝔖 Bobbio Scriptorium
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Structure-activity relationships of pyrethroid insecticides. Part 2. The use of molecular dynamics for conformation searching and average parameter calculation

✍ Scribed by Brian D. Hudson; Ashley R. George; Martyn G. Ford; David J. Livingstone


Publisher
Springer Netherlands
Year
1992
Tongue
English
Weight
559 KB
Volume
6
Category
Article
ISSN
0920-654X

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✦ Synopsis


Molecular dynamics simulations have been performed on a number of conformationally flexible pyrethroid insecticides. The results indicate that molecular dynamics is a suitable tool for conformational searching of small molecules given suitable simulation parameters. The structures derived from the simulations are compared with the static conformation used in a previous study. Various physicochemical parameters have been calculated for a set of conformations selected from the simulations using multivariate analysis. The averaged values of the parameters over the selected set (and the factors derived from them) are compared with the single conformation values used in the previous study.