## Abstract A short and efficient protocol for the asymmetric synthesis of __cis__‐ and __trans__‐3,4‐dihydro‐2,4,8‐trihydroxynaphthalen‐1(2__H__)‐one (**1** and **2**, resp.) is described, with a phthalide annulation as the key step. Introduction of a OH substituent at position 2 was performed by
Stereocontrolled synthesis of enantiopure cis- and trans-3,4,4a,5,8,8a-hexahydro-1H-quinolin-2-ones
✍ Scribed by Mercedes Amat; Maria Pérez; Annamaria T. Minaglia; Daniele Passarella; Joan Bosch
- Book ID
- 108284393
- Publisher
- Elsevier Science
- Year
- 2008
- Tongue
- English
- Weight
- 200 KB
- Volume
- 19
- Category
- Article
- ISSN
- 0957-4166
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