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Simple preparation of a useful C/D-ring fragment for the construction of 11-keto steroids

✍ Scribed by Gilbert Stork; Glenn Clark; Thomas Weller

Publisher: Elsevier Science
Year: 1984
Tongue: French
Weight: 189 KB
Volume: 25
Category: Article
ISSN: 0040-4039
DOI: 10.1016/s0040-4039(01)91285-7

No coin nor oath required. For personal study only.

✦ Synopsis

Starting with the readily available enol-lactone 2 the indanonepropionic acid J_ is prepared in few steps with 33% overall yield, We have recently shown that 11-keto steroids ( e.g. k ) can be construc-

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