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Selective Mechanism-Based Inactivation of CYP3A4 by CYP3cide (PF-04981517) and Its Utility as an In Vitro Tool for Delineating the Relative Roles of CYP3A4 versus CYP3A5 in the Metabolism of Drugs

✍ Scribed by Walsky, R. L.; Obach, R. S.; Hyland, R.; Kang, P.; Zhou, S.; West, M.; Geoghegan, K. F.; Helal, C. J.; Walker, G. S.; Goosen, T. C.; Zientek, M. A.

Book ID: 121876113
Publisher: American Society for Pharmacology and Experimental Therapeutics
Year: 2012
Tongue: English
Weight: 459 KB
Volume: 40
Category: Article
ISSN: 0090-9556
DOI: 10.1124/dmd.112.045302

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